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Synthesis and in vitro evaluation of new fluorinated quinoline derivatives with high affinity for PDE5: Towards the development of new PET neuroimaging probes
Jianrong Liu
,
Aurelie Maisonial-Besset
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Barbara Wenzel
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Damien Canitrot
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Ariane Baufond
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et al.
Journal articles
hal-01671041v1
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Bis-14-membered ring diketal diamines: Synthesis and evaluation of their anti-HIV and anti-tumoral activities.
Radouane Affani
,
Franck Pélissier
,
Anne-Marie Aubertin
,
Denise Dugat
Journal articles
hal-00384465v1
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Improved potency of pyridin-2(1H)one derivatives for the treatment of mechanical allodynia
Alexia Visseq
,
Amélie Descheemaeker
,
Karine Hérault
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Francis Giraud
,
Isabelle Abrunhosa-Thomas
,
et al.
Journal articles
hal-03334145v1
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Synthesis and biological activities of aminopyrimidyl-indoles structurally related to meridianins
Rufine Akué-Gédu
,
Eric Debiton
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Yoan Ferandin
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Laurent Meijer
,
Michelle Prudhomme
,
et al.
Bioorganic and Medicinal Chemistry, 2009, 17, pp.4420-4424
Journal articles
hal-00392799v1
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Synthesis and biological evaluation of diversely substituted indolin-2-ones
Fadoua Bouchikhi
,
Emilie Rossignol
,
Martine Sancelme
,
Bettina Aboab
,
Fabrice Anizon
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et al.
European Journal of Medicinal Chemistry, 2008, 43, pp.2316-2322
Journal articles
hal-00333575v2
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Stereoselective Synthesis of Fluorinated Galactopyranosides as Potential Molecular Probes for Galactophilic Proteins: Assessment of Monofluorogalactoside–LecA Interactions
Vincent Denavit
,
Danny Lainé
,
Chahrazed Bouzriba
,
Elena Shanina
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Emilie Gillon
,
et al.
Journal articles
hal-02104563v1
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A Novel HPLC Method for Direct Detection of Nitric Oxide Scavengers from Complex Plant Matrices and Its Application to Aloysia triphylla Leaves
Didier Fraisse
,
Alexandra Degerine-Roussel
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Alexis Bred
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Samba Ndoye
,
Magali Vivier
,
et al.
Journal articles
hal-01873226v1
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A Photochemical Approach to Pyridopyrroloquinoline Derivatives as New Potential Anticancer Agents
Pierre-Jean Aragon
,
Ange-Désiré Yapi
,
Frédéric Pinguet
,
Jean-Michel Chezal
,
Jean-Claude Teulade
,
et al.
Journal articles
hal-02384520v1
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Gliotransmission and Brain Glucose Sensing: Critical Role of Endozepines
Damien Lanfray
,
Sébastien Arthaud
,
Johanne Ouellet
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Vincent Compère
,
Jean-Luc Do Rego
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et al.
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hal-01962799v1
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Benefits of the ipowder® extraction process applied to Melissa officinalis L.: improvement of antioxidant activity and in vitro gastro-intestinal release profile of rosmarinic acid
Valérie Bardot
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Anaïs Escalon
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Isabelle Ripoche
,
Sylvain Denis
,
Monique Alric
,
et al.
Journal articles
hal-02441644v1
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A proof of principle study using radiopharmaceuticals to quantify and localize container-content interactions in medical syringes
C. Dupire
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P. Chennell
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B. Pereira
,
N. Courtiol
,
S. Buj
,
et al.
Journal articles
hal-04144593v1
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Synthesis and biological evaluation of Haspin inhibitors: kinase inhibitory potency and cellular activity
Wael Zeinyeh
,
Yannick Esvan
,
Béatrice Josselin
,
Mathilde Defois
,
Blandine Baratte
,
et al.
Journal articles
hal-03764791v1
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Heteropolysaccharides from S. cerevisiae show anti-adhesive properties against E. coli associated with Crohn’s disease
Adeline Sivignon
,
Shin-Yi Yu
,
Nathalie Ballet
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Pascal Vandekerckove
,
Nicolas Barnich
,
et al.
Journal articles
hal-03373401v1
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Effect of proteases against biofilms of Staphylococcus aureus and Staphylococcus epidermidis
Pierre-Henri Elchinger
,
C. Delattre
,
S. Faure
,
O. Roy
,
S. Badel
,
et al.
Journal articles
hal-01081362v1
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Metabolic and Anti-Inflammatory Protective Properties of Human Enriched Serum Following Artichoke Leaf Extract Absorption: Results from an Innovative Ex Vivo Clinical Trial
Fabien Wauquier
,
Line Boutin-Wittrant
,
Aurélien Viret
,
Laure Guilhaudis
,
Hassan Oulyadi
,
et al.
Journal articles
hal-03326084v1
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Pharmacological characterization of (4R)-alkyl glutamate analogues at the ionotropic glutamate receptors - Focus on subtypes iGluR5-7
Lennart Bunch
,
Thierry Gefflaut
,
Sébastien Alaux
,
Emmanuelle Sagot
,
Brigitte Nielsen
,
et al.
European Journal of Pharmacology, 2009, 609, pp.1-4
Journal articles
hal-00376953v1
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Synthesis, in vitro antiproliferative activities, and Chk1 inhibitory properties of pyrrolo[3,4-a]carbazole-1,3-diones, pyrrolo[3,4-c]carbazole-1,3-diones, and 2-aminopyridazino[3,4-a]pyrrolo[3,4-c]carbazole-1,3,4,7-tetraone
Elisabeth Conchon
,
Fabrice Anizon
,
Bettina Aboab
,
Roy Golsteyn
,
Stéphane Leonce
,
et al.
European Journal of Medicinal Chemistry, 2008, 43, pp.282-292
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hal-00255899v1
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Chemo-enzymatic synthesis of a series of 2,4-syn-functionalized (S)-glutamate analogues: new insight into the structure-activity relation of ionotropic glutamate receptor subtypes 5, 6, and 7.
Emmanuelle Sagot
,
Darryl S. Pickering
,
Xiasui Pu
,
Michelle Umberti
,
Tine B. Stensbol
,
et al.
Journal of Medicinal Chemistry, 2008, 51, pp.4093-4103
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hal-00323861v1
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Current Opinion on Chitosan and its Derivatives: Biological Impact in Antimicrobial Applications From Nature to Chitosan and It Derivatives: How it is Working?
Cédric Delattre
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hal-01657856v1
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Synthesis and biological evaluation of new dipyrrolo[3,4-a:3,4-c]carbazole-1,3,4,6-tetraones, substituted with various saturated and unsaturated side chains via palladium catalyzed cross-coupling reactions
Hélène Henon
,
Fabrice Anizon
,
Roy Golsteyn
,
Stéphane Leonce
,
Robert Hofmann
,
et al.
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hal-00023499v1
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Synthesis and in Vitro Cytotoxic Evaluation of New Derivatives of Pyrido[1,2-a]benzimidazolic Ring System: The Pyrido[1,2:1,2]imidazo[4,5-h]quinazolines
Marianne Dupuy
,
Frédéric Pinguet
,
Olivier Chavignon
,
Jean-Michel Chezal
,
Jean-Claude Teulade
,
et al.
Journal articles
hal-02384513v1
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Chemo-enzymatic synthesis of (2S,4R)-2-amino-4-(3-(2,2-diphenylethylamino)-3 oxopropyl)pentanedioic acid: A novel Selective inhibitor of human excitatory amino acid transporter subtype 2
Emmanuelle Sagot
,
Anders A. Jensen
,
Darryl S. Pickering
,
Xiasui Pu
,
Michelle Umberti
,
et al.
Journal of Medicinal Chemistry, 2008, 51, pp.4085-4092
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hal-00323786v1
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A three-step synthesis from rebeccamycin of an efficient checkpoint kinase 1 inhibitor.
Fabrice Anizon
,
Roy Golsteyn
,
Stéphane Leonce
,
Bruno Pfeiffer
,
Michelle Prudhomme
European Journal of Medicinal Chemistry, 2009, 44, pp.2234-2238
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hal-00371170v1
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Development of a new radiofluorinated quinoline analog for PET imaging of phosphodiesterase 5 (PDE5) in brain
Jianrong Liu
,
Barbara Wenzel
,
Sladjana Dukic-Stefanovic
,
Rodrigo Teodoro
,
Friedrich-Alexander Ludwig
,
et al.
Journal articles
hal-01677542v1
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Synthesis and Biological Evaluation of Indoloquinolines and Pyridocarbazoles: A New Example of Unexpected Photoreduction Accompanying Photocyclization
Pierre-Jean Aragon
,
Ange-Désiré Yapi
,
Frédéric Pinguet
,
Jean-Michel Chezal
,
Jean-Claude Teulade
,
et al.
Journal articles
hal-02384499v1
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Neuroprotective Effects of a Novel Demeclocycline Derivative Lacking Antibiotic Activity: From a Hit to a Promising Lead Compound
Rodrigo Tomas-Grau
,
Florencia González-Lizárraga
,
Diego Ploper
,
César Avila
,
Sergio Socías
,
et al.
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hal-03775634v1
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Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitors.
Rajâa Boulahjar
,
Aziz Ouach
,
Stéphane Bourg
,
Pascal Bonnet
,
Olivier Lozach
,
et al.
Journal articles
hal-01212495v1
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Quick and Simple Detection Technique to Assess the Binding of Antimicrotubule Agents to the Colchicine-Binding Site
Sébastien Fortin
,
Jacques Lacroix
,
Marie-France Côté
,
Emmanuel Moreau
,
Éric Petitclerc
,
et al.
Journal articles
hal-01677569v1
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Azoliums and Ag(I)‐N‐Heterocyclic Carbene Thioglycosides: Synthesis, Reactivity and Bioactivity
Dmytro Ryzhakov
,
Audrey Beillard
,
Franck Le Bideau
,
Riyadh Ahmed Atto Al‐shuaeeb
,
Mouad Alami
,
et al.
Journal articles
hal-03648181v2
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Synthesis, chekpoint kinase 1 inhibitory properties and in vitro antiproliferative activities of new pyrrolocarbazoles
Elisabeth Conchon
,
Fabrice Anizon
,
Bettina Aboab
,
Roy Golsteyn
,
Stéphane Leonce
,
et al.
Bioorganic and Medicinal Chemistry, 2008, 16, pp.4419-4430
Journal articles
hal-00277522v1
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